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VPC-13163

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Purity:97.24%

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COA HPLC HNMR

VPC-13163

Catalog No. T29110Cas No. 6637-10-1

VPC-13163 (NSC-52361) has strong anti-proliferative activity against LNCaP and Enzalutamide-resistant prostate cancer cell lines (MR49F) whereas it did not affect the growth of AR independent PC3 cell line. It also inhibits Prostate Specific Antigen (PSA) in both LNCaP and MR49F and reduces expression of AR target genes, PSA and TMPRSS2. These findings suggest that VPC-13566 exhibits AR BF3 specific mechanism of action.

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Pack Size	Price	Availability
1 mg	$137	In Stock
5 mg	$336	In Stock
10 mg	$497	In Stock
25 mg	$793	In Stock
50 mg	$1,130	In Stock
100 mg	$1,520	In Stock
500 mg	$2,970	In Stock
1 mL x 10 mM (in DMSO)	$295	In Stock

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Product Introduction

Bioactivity

Description

Alias

2,3-dihydro-2,3'-Bi-1H-indole, VPC13163, NSC52361, NSC 52361, VPC 13163

Chemical Properties

Molecular Weight	234.3
Formula	C16H14N2
Cas No.	6637-10-1

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 65 mg/ml (277.42 mM)

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	4.2680 mL	21.3402 mL	42.6803 mL	213.4016 mL
5 mM	0.8536 mL	4.2680 mL	8.5361 mL	42.6803 mL
10 mM	0.4268 mL	2.1340 mL	4.2680 mL	21.3402 mL
20 mM	0.2134 mL	1.0670 mL	2.1340 mL	10.6701 mL
50 mM	0.0854 mL	0.4268 mL	0.8536 mL	4.2680 mL
100 mM	0.0427 mL	0.2134 mL	0.4268 mL	2.1340 mL

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