Shopping Cart
- Remove All
Your shopping cart is currently empty
(RS)-Butyryltimolol
😃Good
Catalog No. T13439Cas No. 2320274-78-8
(RS)-Butyryltimolol, the racemate of Butyryltimolol, is an effective prodrug of Timolol that improves corneal penetration and acts as a β-adrenergic blocker [1][2].
(RS)-Butyryltimolol
😃Good
Catalog No. T13439Cas No. 2320274-78-8
(RS)-Butyryltimolol, the racemate of Butyryltimolol, is an effective prodrug of Timolol that improves corneal penetration and acts as a β-adrenergic blocker [1][2].
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 2 mg | $61 | 5 days |
Bulk & Custom
Add to Cart
Questions
View MoreInhibitors Related to "(RS)-Butyryltimolol"
Esomeprazole
T20626119141-88-7
Esomeprazole is the S-isomer of omeprazole, inhibits the lysosomal cysteine protease legumain to prevent cancer metastasis. Esomeprazole is a proton pump inhibitors (PPI).
- $57
Size
QTY
N-Ethylmaleimide
Cited
NEM, Ethylmaleimide, 1-Ethyl-1H-pyrrole-2,5-dione
T3088128-53-0
N-Ethylmaleimide (NEM) is a reagent for alkylation of free sulfhydryl groups, a cysteine protease inhibitor used in experimental biochemistry. N-Ethylmaleimide is also a deubiquitinating enzyme inhibitor that specifically inhibits phosphate transport in mitochondria.
- $39
Size
QTY
Cited2-Aminoethanethiol
β-Mercaptoethylamine, β-MEA, Cysteamine, 2-Mercaptoethylamine
T108060-23-1
2-Aminoethanethiol (Cysteamine) is a Cystine Depleting Agent. The mechanism of action of cysteamine is as a Cystine Disulfide Reduction.
- $45
Size
QTY
KGP94
KGP-94, KGP 94
T277301131456-28-4
KGP94 is an inhibitor of cysteine protease Cathepsin L(CTSL).
- $115
Size
QTY
Leupeptin Hemisulfate
Cited
T6564103476-89-7
Leupeptin hemisulfate is a protease inhibitor with cell membrane-permeable, reversible, competitive, and oral activities. Leupeptin hemisulfate inhibits the activity of Cathepsin B, Cathepsin H, and Cathepsin L, and blocks fusion of amphipathic lysosomes. Leupeptin hemisulfate also has anti-inflammatory activity.
- $47
Size
QTY
CitedPapain
T195039001-73-4
Papain, a cysteine protease of the peptidase C1 family, is utilized in the food, pharmaceutical, textile, and cosmetic industries.
- $45
Size
QTY
PMSF Cited
Phenylmethylsulfonyl fluoride, Benzylsulfonyl fluoride
T0789329-98-6
Phenylmethanesulfonyl fluoride (PMSF (Phenylmethylsulfonyl fluoride)) is an enzyme inhibitor that inactivates IRC-50 arvin, subtilisin, and the fatty acid synthetase complex.
- $33
Size
QTY
CitedZ-Lys-OH
T658682212-75-1
Z-Lys-OH is a competitive inhibitor of papain, a lysine derivative.
- $29
Size
QTY
2-Cyanopyrimidine
2-cyano-Pyrimidine
T745114080-23-0
2-Cyanopyrimidine (m-Hydroxyphenylpropionic acid) is inhibitor of cathepsin K(IC50 : 170 nM)
- $29
Size
QTY
E-64 Cited
Proteinase inhibitor E 64, E64, E 64
T603766701-25-5
E-64 (Proteinase inhibitor E 64) is an irreversible and specific inhibitor of cysteine proteases, exhibiting an IC50 of 9 nM for papain.
- $31
Size
QTY
Cited(S)-(+)-Ibuprofen
Dexibuprofen, (S)-Ibuprofen
T044851146-56-6
(S)-(+)-Ibuprofen (Dexibuprofen) , is a non-steroidal anti-inflammatory drug (NSAID), inhibiting cyclooxygenase (COX).
- $35
Size
QTY
Aloxistatin Cited
Loxistatin, E64d, E64c ethyl ester
T604088321-09-9
Aloxistatin (E64d) is an inhibitor of cysteine protease with blood platelet aggregation inhibiting activity. Aloxistatin is an irreversible, membrane-permeable inhibitor of lysosomal and cytosolic cysteine proteases with the ability to inhibit calpain activity in intact platelets.
- $36
Size
QTY
CitedContact us for more batch information
Resource Download
Product Introduction
Bioactivity
Chemical Properties
| Description | (RS)-Butyryltimolol, the racemate of Butyryltimolol, is an effective prodrug of Timolol that improves corneal penetration and acts as a β-adrenergic blocker [1][2]. |
| In vitro | Butyryltimolol is a prodrug of Timolol. Butyryltimolol is equally effective as 240-min nasolacrimal blockade in enhancing ocular drug absorption [1]. |
| Molecular Weight | 386.51 |
| Formula | C17H30N4O4S |
| Cas No. | 2320274-78-8 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 100 mg/mL (258.73 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
| ||||||||||||||||||||||||||||||||||||
Calculator
In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
Dose Conversion
You can also refer to dose conversion for different animals. More Dose Conversion
Tech Support
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
Preview
Related Tags: buy (RS)-Butyryltimolol | purchase (RS)-Butyryltimolol | (RS)-Butyryltimolol cost | order (RS)-Butyryltimolol | (RS)-Butyryltimolol chemical structure | (RS)-Butyryltimolol in vitro | (RS)-Butyryltimolol formula | (RS)-Butyryltimolol molecular weight
- TOP
Feedback
Hello! How can I help you today? 
Copyright © 2015-2024 TargetMol Chemicals Inc. All Rights Reserved.