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β-Endorphin (1-27) (human) acetate

Catalog No. T38193L

Synonyms: β-Endorphin (1-27) (human) acetate(76622-84-9 Free base)

β-Endorphin (1-27) (human) acetate, existing in the hypophysis cerebri and hypothalamus, exhibits antinociception activity. β-Endorphin (1-27) (human) acetate is an agonist of opioid receptor, showing preferred affinity for μ-opioid receptor and δ-opioid

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β-Endorphin (1-27) (human) acetate Chemical Structure

β-Endorphin (1-27) (human) acetate, CAS N/A

Pack Size	Availability	Price/USD
1 mg	In stock	$ 195.00
5 mg	In stock	$ 437.00
10 mg	In stock	$ 646.00
25 mg	In stock	$ 987.00
50 mg	In stock	$ 1,380.00
100 mg	In stock	$ 1,860.00

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Purity: 96.52%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

In vitro

β-Endorphin (1-27) (human) acetate inhibits the conduction of pain and agitation of nociceptors to exert an analgesic effect. β-Endorphin (1-27) (human) acetate combines together with the opioid receptors in hyperalgesia. β-Endorphin (1-27) (human) acetate suppresses the release of substance P at the level of spinal cord and blocks the conduction of pain on the primary sensory neurons. β-Endorphin (1-27) (human) acetate activates the endogenous analgesia system located in the CNS[1].

Synonyms	β-Endorphin (1-27) (human) acetate(76622-84-9 Free base)
Molecular Weight	3082.52
Formula	C141H221N33O42S

Storage

keep away from moisture

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Luan YH, et al. Action of β-endorphin and nonsteroidal anti-inflammatory drugs, and the possible effects of nonsteroidal anti-inflammatory drugs on β-endorphin. J Clin Anesth. 2017 Feb;37:123-128. 2. Narita M, et al. Evidence for the existence of the beta-endorphin-sensitive "epsilon-opioid receptor" in the brain: the mechanisms of epsilon-mediated antinociception. Jpn J Pharmacol. 1998 Mar;76(3):233-53.

Related compound libraries

This product is contained In the following compound libraries：

Bioactive Compound Library Peptide Compound Library Bioactive Compounds Library Max

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Keywords

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