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4-Hydroxymephenytoin
🥰Excellent
Catalog No. T10147Cas No. 61837-65-8
Alias (+/-)-4'-Hydroxymephenytoin
4-Hydroxymephenytoin ((+/-)-4'-Hydroxymephenytoin) is the metabolism of an antiepileptic drug mephenytoin. Mephenytoin is used as a CYP2C19 substrate.
4-Hydroxymephenytoin
🥰Excellent
Purity: 99.58%
Catalog No. T10147Alias (+/-)-4'-HydroxymephenytoinCas No. 61837-65-8
4-Hydroxymephenytoin ((+/-)-4'-Hydroxymephenytoin) is the metabolism of an antiepileptic drug mephenytoin. Mephenytoin is used as a CYP2C19 substrate.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $39 | In Stock | |
| 5 mg | $72 | In Stock | |
| 10 mg | $113 | In Stock | |
| 25 mg | $228 | In Stock | |
| 50 mg | $372 | In Stock | |
| 100 mg | $597 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $97 | In Stock |
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Purity:99.58%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | 4-Hydroxymephenytoin ((+/-)-4'-Hydroxymephenytoin) is the metabolism of an antiepileptic drug mephenytoin. Mephenytoin is used as a CYP2C19 substrate. |
| In vitro | 4-Hydroxymephenytoin, a metabolite of the antiepileptic drug mephenytoin, serves as a CYP2C19 substrate[1]. It is utilized in the development of UltraPerformance LC (UPLC) tandem mass spectrometry assays to assess CYP probe drugs and their pertinent metabolites in human urine or plasma samples[2]. |
| Alias | (+/-)-4'-Hydroxymephenytoin |
| Molecular Weight | 234.25 |
| Formula | C12H14N2O3 |
| Cas No. | 61837-65-8 |
| Smiles | CCC1(NC(=O)N(C)C1=O)c1ccc(O)cc1 |
| Relative Density. | 1.249 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 90 mg/mL (384.2 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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