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BMS986299

Catalog No. T9572 CAS 2242952-69-6

BMS986299 is a modulator of NLRP3 with an EC50 of 1.28 μM and can be used in studies about NLRP3 signaling and the treatment of associated diseases.

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BMS986299, CAS 2242952-69-6

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Purity: 98%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

BMS986299 is a modulator of NLRP3 with an EC50 of 1.28 μM and can be used in studies about NLRP3 signaling and the treatment of associated diseases.

Molecular Weight	349.398
Formula	C18H19N7O
CAS No.	2242952-69-6

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

DMSO: 30 mg/mL (85.86 mM), Need ultrasonic

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Gary Glick, et al. Substituted imidazo-quinolines as nlrp3 modulators. WO2018152396A1.

Related Products

Related compounds with same targets

Emlenoflast Asymmetric dimethylarginine 6-Biopterin NLRP3-IN-10 L-Canavanine sulfate CY-09 MCC950 Imperatorin

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

BMS986299 2242952-69-6 NF-Κb Immunology/Inflammation NOD Inhibitor inhibitor inhibit

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.