Powder: -20°C for 3 years | In solvent: -80°C for 1 year
ERRγ Inverse Agonist 1 (Compound 12) is a potent, selective and orally bioavailable Estrogen-related Receptor grammar (ERRγ) inverse agonist (IC 50=40 nM) [1].
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 6-8 weeks | $ 1,520.00 | |
50 mg | 6-8 weeks | $ 1,980.00 | |
100 mg | 6-8 weeks | $ 2,500.00 |
Description | ERRγ Inverse Agonist 1 (Compound 12) is a potent, selective and orally bioavailable Estrogen-related Receptor grammar (ERRγ) inverse agonist (IC 50=40 nM) [1]. |
Targets&IC50 | ERRβ:1.330 μM, ERα:1.240 μM, ERRγ:0.040 μM |
Molecular Weight | 529.54 |
Formula | C30H38Cl2N2O2 |
CAS No. | 2316832-86-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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ERRγ Inverse Agonist 1 2316832-86-5 Endocrinology/Hormones Estrogen/progestogen Receptor ERRgamma Inverse Agonist 1 ERRr Inverse Agonist 1 inhibitor inhibit