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S1PR1 modulator 1
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S1PR1 modulator 1
Catalog No. T12821Cas No. 2328109-05-1
S1PR1 modulator 1 is a selective inhibitor of S1PR1 with a pIC50 of 7.6.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $59 | In Stock | |
| 5 mg | $122 | In Stock | |
| 10 mg | $173 | In Stock | |
| 25 mg | $285 | In Stock | |
| 50 mg | $422 | In Stock | |
| 100 mg | $626 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $141 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | S1PR1 modulator 1 is a selective inhibitor of S1PR1 with a pIC50 of 7.6. |
| In vitro | S1PR1 modulator 1 shows >40- and >80-fold selectivity, over the other S1PR isoforms S1PR3 (pIC50, 6), S1PR2 and S1PR4 (pIC50s, <5)[1]. |
| Molecular Weight | 408.51 |
| Formula | C23H24N2O3S |
| Cas No. | 2328109-05-1 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | ||||||||||||||||||||
| Solubility Information | DMSO: 6.11 mg/mL (14.96 mM)  | ||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||
DMSO
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