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SYM 2081

Catalog No. T16963 CAS 31137-74-3

SYM 2081 is a specific kainate receptor agonist with an IC50 value of 35 nM for [3H]-kainate binding. SYM 2081 depolarizes the muscle and reduces the EPSP amplitude.

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SYM 2081, CAS 31137-74-3

Pack Size	Availability	Price/USD
1 mg	In stock	$ 87.00
5 mg	In stock	$ 213.00
10 mg	In stock	$ 313.00
25 mg	In stock	$ 533.00
50 mg	In stock	$ 768.00
100 mg	In stock	$ 1,080.00
500 mg	In stock	$ 2,160.00

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Purity: 99.59%

Biological Description

Chemical Properties

Storage & Solubility Information

Description	SYM 2081 is a specific kainate receptor agonist with an IC50 value of 35 nM for [3H]-kainate binding. SYM 2081 depolarizes the muscle and reduces the EPSP amplitude.
Targets&IC50	Kainate receptor:35 nM

Molecular Weight	161.16
Formula	C6H11NO4
CAS No.	31137-74-3

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

H2O: 45.0 mg/mL (279.2 mM), Sonification is recommended.

References and Literature

1. Lee JY, et al. Furthering pharmacological and physiological assessment of the glutamatergic receptors at the Drosophila neuromuscular junction. Comp Biochem Physiol C Toxicol Pharmacol. 2009 Nov;150(4):546-57.

Related compound libraries

This product is contained In the following compound libraries：

Bioactive Compound Library Neuronal Signaling Compound Library Bioactive Compounds Library Max

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

SYM 2081 31137-74-3 Membrane transporter/Ion channel Neuroscience iGluR SYM-2081 SYM2081 inhibitor inhibit

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