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AR-08
🥰Excellent
Catalog No. T10052Cas No. 226081-74-9
AR-08 is a potent α2-adrenergic receptor agonist for the study of ADHD and attention deficit.
AR-08
🥰Excellent
Purity: 99.7%
Catalog No. T10052Cas No. 226081-74-9
AR-08 is a potent α2-adrenergic receptor agonist for the study of ADHD and attention deficit.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | 665 € | In Stock | |
| 5 mg | 1.710 € | In Stock |
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Purity:99.7%
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With extensive experience in compound synthesis, we can provide rapid custom synthesis services for this product according to your research needs.Product Introduction
Bioactivity
Chemical Properties
| Description | AR-08 is a potent α2-adrenergic receptor agonist for the study of ADHD and attention deficit. |
| In vivo | After intravenous administration of a single dose of 15 mg/kg to 6 healthy lactating goats, the pharmacokinetic behavior of Ibafloxacin is studied. Plasma concentrations of Ibafloxacin are determined by high-performance liquid chromatography with fluorescence detection. Following intravenous injection, Ibafloxacin exhibits very rapid initial distribution, with a mean half-life of 0.35 h, followed by slower elimination, with a mean half-life of 3.76 h. The elimination half-life of Ibafloxacin after oral administration has been reported to be 3.83 h in dogs and 3.00 h in cats[1]. |
| Molecular Weight | 240.26 |
| Formula | C12H12N6 |
| Cas No. | 226081-74-9 |
| Smiles | N#CC=1C=C(NC2=NCCN2)C(=C3N=CNC13)C |
| Relative Density. | 1.50 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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