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BJJF078

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Purity:98.19%

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COA HPLC HNMR

BJJF078

Catalog No. T67865Cas No. 2531244-56-9

BJJF078, an aminopiperidine derivative, is a potent inhibitor of recombinant human and mouse glutamine aminotransferase (TG2) activity, with IC50 values of 41 and 54 nM for human and mouse glutamine aminotransferase, respectively.BJJF078 inhibits TG1 enzyme, with an IC50 of 0.16 μM.BJJF078 can be used to study multiple sclerosis (MS). BJJF078 can be used to study multiple sclerosis (MS).

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Pack Size	Price	Availability
1 mg	$53	In Stock
5 mg	$111	In Stock
10 mg	$159	In Stock
25 mg	$266	In Stock
50 mg	$396	In Stock
100 mg	$589	In Stock

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Product Introduction

Bioactivity

Description	BJJF078, an aminopiperidine derivative, is a potent inhibitor of recombinant human and mouse glutamine aminotransferase (TG2) activity, with IC50 values of 41 and 54 nM for human and mouse glutamine aminotransferase, respectively.BJJF078 inhibits TG1 enzyme, with an IC50 of 0.16 μM.BJJF078 can be used to study multiple sclerosis (MS). BJJF078 can be used to study multiple sclerosis (MS).
Targets&IC50	TGase 1:0.16 μM, TG2 (human):41 nM, TG2 (mouse):54 nM

Chemical Properties

Molecular Weight	523.6
Formula	C27H29N3O6S
Cas No.	2531244-56-9

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

Solubility Information

DMSO: 60 mg/mL (114.59 mM)

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	1.9099 mL	9.5493 mL	19.0985 mL	95.4927 mL
5 mM	0.3820 mL	1.9099 mL	3.8197 mL	19.0985 mL
10 mM	0.1910 mL	0.9549 mL	1.9099 mL	9.5493 mL
20 mM	0.0955 mL	0.4775 mL	0.9549 mL	4.7746 mL
50 mM	0.0382 mL	0.1910 mL	0.3820 mL	1.9099 mL
100 mM	0.0191 mL	0.0955 mL	0.1910 mL	0.9549 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

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A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc