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CV-6209
CV-6209 is a potent antagonist of the platelet-activating factor (PAF) receptor.
Catalog No. T27102Cas No. 100488-87-7
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Purity:100%
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CV-6209
Catalog No. T27102Alias CV6209, CV 6209Cas No. 100488-87-7
CV-6209 is a potent antagonist of the platelet-activating factor (PAF) receptor.
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Product Introduction
Bioactivity
Chemical Properties
| Description | CV-6209 is a potent antagonist of the platelet-activating factor (PAF) receptor. |
| In vitro | CV-6209 (0.2-2 μM; pretreatment for 30 min) inhibited PAF-induced degranulation of LAD2 and hLMC MC; CV-6209 (30 nM) inhibited the release of [3H]5-hydroxytryptamine from rabbit platelets stimulated by PAF [4]. |
| In vivo | CV-6209 (i.v.) inhibited PAF (0.3 μg/kg; i.v.) induced hypotension in rats (ED50=0.009 mg/kg) but had no effect on arachidonic acid, histamine, bradykinin and isobarbital-induced hypotension [4]. CV-6209 (66 μg; i.v.) reduced asparaginase-induced hypersensitivity compared to untreated sensitized mice [5]. |
| Alias | CV6209, CV 6209 |
| Molecular Weight | 642.31 |
| Formula | C34H60ClN3O6 |
| Cas No. | 100488-87-7 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 80 mg/mL (124.55 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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