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Eltenac
🥰Excellent
Catalog No. T27254Cas No. 72895-88-6
Alias BY-820, BY820, BY 820, B-78820, B78820, B 78820
Eltenac (B78820) is a non-steroidal anti-inflammatory, COX inhibitor with analgesic activity.Eltenac inhibits COX-1 and COX-2 and is used in the study of Acute Respiratory Distress Syndrome (ARDS).
Eltenac
🥰Excellent
Purity: 98.78%
Catalog No. T27254Alias BY-820, BY820, BY 820, B-78820, B78820, B 78820Cas No. 72895-88-6
Eltenac (B78820) is a non-steroidal anti-inflammatory, COX inhibitor with analgesic activity.Eltenac inhibits COX-1 and COX-2 and is used in the study of Acute Respiratory Distress Syndrome (ARDS).
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 500 μg | $383 | In Stock | |
| 1 mg | $725 | In Stock | |
| 5 mg | $2,270 | In Stock |
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Purity:98.78%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Eltenac (B78820) is a non-steroidal anti-inflammatory, COX inhibitor with analgesic activity.Eltenac inhibits COX-1 and COX-2 and is used in the study of Acute Respiratory Distress Syndrome (ARDS). |
| Targets&IC50 | COX-2:0.03 μM, COX-1:0.03 μM |
| In vitro | Eltenac is the most potent inhibitor of the COX-2 isomer (IC50 = 0.02 lM), although there is a significant difference between the two COX isomers (P = 0.0014) and the efficacy ratio is 4.80, but the inhibitory effect of Eltenac on COX-2 isomers is still strong. [5] |
| In vivo | Etinac (10 mg/kg; oral; female Sprague-Dawley rats, 150-190 lbs; rat paw edema model) was effective in reducing paw volume increase by 52% [1]. |
| Alias | BY-820, BY820, BY 820, B-78820, B78820, B 78820 |
| Molecular Weight | 302.18 |
| Formula | C12H9Cl2NO2S |
| Cas No. | 72895-88-6 |
| Smiles | O=C(O)CC1=CSC=C1NC=2C(Cl)=CC=CC2Cl |
| Relative Density. | 1.539g/cm3 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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