Shopping Cart

Remove All
Your shopping cart is currently empty

GCN2-IN-1

Name: GCN2-IN-1
Brand: TargetMol
SKU: T11373
Price: 67 USD
Availability: InStock
Rating: 5 (10 reviews)

GCN2-IN-1 (A-92) is an effective GCN2 inhibitor and can be utilized in cancer research as a chemotherapeutic agent.

Catalog No. T11373Cas No. 1448693-69-3

Select Batch

Purity:99.45%

Resource Download

COA HNMR HPLC

GCN2-IN-1

Catalog No. T11373Cas No. 1448693-69-3

GCN2-IN-1 (A-92) is an effective GCN2 inhibitor and can be utilized in cancer research as a chemotherapeutic agent.

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Pack Size	Price	Availability
1 mg	$67	In Stock
5 mg	$147	In Stock
10 mg	$228	In Stock
25 mg	$478	In Stock
50 mg	$689	In Stock
100 mg	$982	In Stock
500 mg	$1,960	In Stock
1 mL x 10 mM (in DMSO)	$162	In Stock

Bulk & Custom

Add to Cart

Questions

Related Compound Libraries of "GCN2-IN-1"

Product Introduction

Bioactivity

Description	GCN2-IN-1 (A-92) is an effective GCN2 inhibitor and can be utilized in cancer research as a chemotherapeutic agent.
Targets&IC50	GCN2:<0.3 μM
In vitro	GCN2-IN-1 inhibits GCN2 with an IC50 of <0.3 μM in the enzyme assay and an IC50 of 0.3-3 μM in the cell assay[1].
Alias	A-92

Chemical Properties

Molecular Weight	402.41
Formula	C₁₉H₁₈N₁₀O
Cas No.	1448693-69-3

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

Solubility Information

DMSO: 55 mg/mL (136.68 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.4850 mL	12.4251 mL	24.8503 mL	124.2514 mL
5 mM	0.4970 mL	2.4850 mL	4.9701 mL	24.8503 mL
10 mM	0.2485 mL	1.2425 mL	2.4850 mL	12.4251 mL
20 mM	0.1243 mL	0.6213 mL	1.2425 mL	6.2126 mL
50 mM	0.0497 mL	0.2485 mL	0.4970 mL	2.4850 mL
100 mM	0.0249 mL	0.1243 mL	0.2485 mL	1.2425 mL

Calculator

Molarity Calculator
Dilution Calculator
Reconstitution Calculator
Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

Dose Conversion

You can also refer to dose conversion for different animals. More

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

InhibitorA92GCN2IN1inhibitEukaryotic Initiation Factor (eIF)GCN2 IN 1GCN2-IN-1A 92