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Indirubin Derivative E804 is a potent insulin-like growth factor type 1 receptor (IGF1R) inhibitor with potential antitumor activity.
Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $42 | In Stock | |
5 mg | $92 | In Stock | |
10 mg | $133 | In Stock | |
25 mg | $218 | In Stock | |
50 mg | $325 | In Stock | |
100 mg | $483 | In Stock | |
200 mg | $691 | In Stock | |
1 mL x 10 mM (in DMSO) | $98 | In Stock |
Description | Indirubin Derivative E804 is a potent insulin-like growth factor type 1 receptor (IGF1R) inhibitor with potential antitumor activity. |
Targets&IC50 | CDK2-CyclinE:0.23 μM (EC50), IGF-1R:0.65 μM |
In vitro | Indirubin Derivative E804 is a water-soluble derivative that effectively inhibits insulin-like growth factor 1 receptor (IGF1R) with an IC50 of 0.65 μM. In addition, Indirubin Derivative E804 also inhibits CDK2/CycE with an EC50 of 0.23 μM. [1] |
Molecular Weight | 365.38 |
Formula | C20H19N3O4 |
Cas No. | 854171-35-0 |
Smiles | O=C1NC=2C=CC=CC2C1=C3NC=4C=CC=CC4C3=NOCCC(O)CO |
Relative Density. | 1.44 g/cm3 (Predicted) |
Storage | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
Solubility Information | DMSO: 100 mg/mL (273.69 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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