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KRAS G12C inhibitor 32
Catalog No. T72335Cas No. 2756739-00-9
KRAS G12C Inhibitor 32, an eight-membered heterocyclic compound with nitrogen, acts as a potent inhibitor of KRAS G12C [1].
KRAS G12C inhibitor 32
Catalog No. T72335Cas No. 2756739-00-9
KRAS G12C Inhibitor 32, an eight-membered heterocyclic compound with nitrogen, acts as a potent inhibitor of KRAS G12C [1].
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 25 mg | $1,670 | 8-10 weeks | |
| 50 mg | $2,180 | 8-10 weeks | |
| 100 mg | $2,800 | 8-10 weeks |
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Product Introduction
Bioactivity
Chemical Properties
| Description | KRAS G12C Inhibitor 32, an eight-membered heterocyclic compound with nitrogen, acts as a potent inhibitor of KRAS G12C [1]. |
| In vitro | KRAS G12C inhibitor 32, also known as compound 6 or 7, effectively suppresses the proliferation of NCI-H358IC cells with an IC50 value of 0.015 μM [1]. |
| Molecular Weight | 635.94 |
| Formula | C29H30Cl3FN6O3 |
| Cas No. | 2756739-00-9 |
Storage & Solubility Information
| Storage | Shipping with blue ice. |
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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