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Litorin acetate(55749-97-8 Free base)

Catalog No. T20604L

Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist. It stimulates the contraction of smooth muscle, stimulates gastrin, gastric acid, and pancreatic secretion, and suppresses the nutriment in vivo.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Litorin acetate(55749-97-8 Free base) Chemical Structure

Litorin acetate(55749-97-8 Free base), CAS N/A

Pack Size	Availability	Price/USD
1 mg	In stock	$ 77.00
5 mg	In stock	$ 221.00
10 mg	In stock	$ 356.00
25 mg	In stock	$ 588.00
50 mg	In stock	$ 857.00
100 mg	In stock	$ 1,180.00

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Purity: 97.64%

Biological Description

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Description	Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist. It stimulates the contraction of smooth muscle, stimulates gastrin, gastric acid, and pancreatic secretion, and suppresses the nutriment in vivo.
In vitro	99mTc-Litorin is developed for non-invasive imaging of tumors with overexpressed gastrin-releasing peptide receptors (GRP-R)[1]. [D-Phe1,Leu8,9]Litorin inhibits binding of 125I-[Tyr4] BN to murine Swiss 3T3 cells with a Ki of 5.1 nM[2]. Litorin stimulates 3H-Thymidine incorporation in murine Swiss 3T3 cells with an EC50 of 2.3 nM[2].
In vivo	Litorin stimulates the contraction of smooth muscle, stimulates gastrin, gastric acid, and pancreatic secretion, and suppresses the nutriment in in vivo experiments[2].

Molecular Weight	1145.29
Formula	C53H72N14O13S

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Related compound libraries

This product is contained In the following compound libraries：

GPCR Compound Library Peptide Compound Library Membrane Protein-targeted Compound Library Natural Product Library Natural Product Library for HTS

Related Products

Related compounds with same targets

PD176252 Kuwanon H MK-5046 RC-3095 TFA CD80-IN-3 PD 168368 ML-18 GB-6

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Litorin acetate(55749-97-8 Free base) GPCR/G Protein Bombesin Receptor Litorin acetate inhibitor inhibit

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.