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P32/98 hemifumarate
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P32/98 hemifumarate
Catalog No. T21979Cas No. 251572-86-8
P32/98 hemifumarate is a dipeptidyl peptidase IV (DPP4) inhibitor with hypoglycemic properties that improves insulin sensitivity and β-cell responsiveness in the Zucker diabetic rat model, and may be useful in studies of type 2 diabetes and colitis.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $93 | In Stock | |
| 5 mg | $228 | In Stock | |
| 10 mg | $342 | In Stock | |
| 25 mg | $568 | In Stock | |
| 50 mg | $812 | In Stock | |
| 100 mg | $1,090 | In Stock | |
| 500 mg | $2,180 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | P32/98 hemifumarate is a dipeptidyl peptidase IV (DPP4) inhibitor with hypoglycemic properties that improves insulin sensitivity and β-cell responsiveness in the Zucker diabetic rat model, and may be useful in studies of type 2 diabetes and colitis. |
| In vitro | In porcine proximal tubular cells,P32/98 (hemifumarate) (10 μM; 96 hours) showed no cytotoxicity[2]. |
| In vivo | In Zucker diabetic fatty rats, P32/98 (hemifumarate) (25 mg/kg; oral gavage; once daily) significantly improved glucose tolerance[3]. |
| Alias | P32/98 (hemifumarate)(136259-20-6 free base) |
| Molecular Weight | 520.71 |
| Formula | C22H40N4O6S2 |
| Cas No. | 251572-86-8 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
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