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Pack Size | Price | Availability | Quantity |
---|---|---|---|
5 mg | $64 | In Stock | |
10 mg | $97 | In Stock | |
25 mg | $197 | In Stock | |
50 mg | $328 | In Stock | |
100 mg | $533 | In Stock | |
500 mg | $1,150 | In Stock | |
1 mL x 10 mM (in DMSO) | $64 | In Stock |
Description | PARP10-IN-3 is a potent and selective mono-Adp-ribotransferase PARP10 inhibitor that inhibits human PARP10 (IC50:480 nM). PARP10-IN-3 also inhibited human PARP2 and human PARP15 with IC50 values of 1.7 μM. |
Targets&IC50 | PARP4 (human):7 μM, PARP1 (human):>100 μM, PARP3 (human):>100 μM, PARP2 (human):1.7 μM, PARP15 (human):1.7 μM, TNKS2 (human):6.5 μM, PARP10 (human):480 nM, PARP12 (human):>10 μM, TNKS1(human):21 μM, PARP14 (human):41 μM, PARP16 (human):>10 μM |
In vitro | PARP10-IN-3 exhibits an IC50 of 1-2 μM in HeLa-PARP10 cells as determined by colony formation assay (CFA).[1] |
Molecular Weight | 256.26 |
Formula | C14H12N2O3 |
Cas No. | 2225800-19-9 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||
Solubility Information | DMSO: 9 mg/mL (35.12 mM) ![]() | |||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||
DMSO
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