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SM-6586
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SM-6586
Catalog No. T16897Cas No. 103898-38-0
SM-6586 is a potent calcium channel antagonist with inhibitory effects on Na+/H+ and Na+/Ca2+ exchange channels, and can be used in the study of cerebrovascular disease and hypertension, among other diseases.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $700 | In Stock | |
| 5 mg | $1,800 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | SM-6586 is a potent calcium channel antagonist with inhibitory effects on Na+/H+ and Na+/Ca2+ exchange channels, and can be used in the study of cerebrovascular disease and hypertension, among other diseases. |
| In vivo | In spontaneously hypertensive rats treated with SM-6586, the survival rate after bilateral common carotid artery ligation is higher, the brain water content is lower, and the ATP level is higher, while lactate level is decreased. In focal ischemia models, the SM-treated group shows a reduction of T1 relaxation time. Additionally, the brain water content is significantly decreased in the SM-treated group[1]. |
| Molecular Weight | 489.52 |
| Formula | C26H27N5O5 |
| Cas No. | 103898-38-0 |
| Storage | store at low temperature Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
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