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Y16 acetate(429653-73-6 free base)
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Catalog No. TP2327L
Alias Y16 acetate(53-73-6 free base), ASN-ARG-VAL-TYR-VAL-HIS-PRO-PHE acetate
Y16 acetate(429653-73-6 free base) is a G-protein–coupled Rho GEFs inhibitor; works synergistically with Rhosin/G04 in inhibiting LARG-RhoA interaction, RhoA activation, and RhoA-mediated signaling functions.
Y16 acetate(429653-73-6 free base)
😃Good
Catalog No. TP2327LAlias Y16 acetate(53-73-6 free base), ASN-ARG-VAL-TYR-VAL-HIS-PRO-PHE acetate
Y16 acetate(429653-73-6 free base) is a G-protein–coupled Rho GEFs inhibitor; works synergistically with Rhosin/G04 in inhibiting LARG-RhoA interaction, RhoA activation, and RhoA-mediated signaling functions.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 2 mg | $50 | Backorder | |
| 5 mg | $68 | Backorder | |
| 10 mg | $103 | Backorder | |
| 25 mg | $184 | Backorder | |
| 50 mg | $276 | Backorder | |
| 100 mg | $412 | Backorder |
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Product Introduction
Bioactivity
Chemical Properties
| Description | Y16 acetate(429653-73-6 free base) is a G-protein–coupled Rho GEFs inhibitor; works synergistically with Rhosin/G04 in inhibiting LARG-RhoA interaction, RhoA activation, and RhoA-mediated signaling functions. |
| Alias | Y16 acetate(53-73-6 free base), ASN-ARG-VAL-TYR-VAL-HIS-PRO-PHE acetate |
| Molecular Weight | 1091.24 |
| Formula | C51H74N14O13 |
| Smiles | CC(O)=O.O=C(N[C@@H](CCCNC(N)=N)C(N[C@@H](C(C)C)C(N[C@@H](CC1=CC=C(C=C1)O)C(N[C@@H](C(C)C)C(N[C@@H](CC2=CNC=N2)C(N3[C@@H](CCC3)C(N[C@@H](CC4=CC=CC=C4)C(O)=O)=O)=O)=O)=O)=O)=O)[C@H](CC(N)=O)N |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||
| Solubility Information | DMSO: 10 mM | ||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||
DMSO
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For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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