store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 700.00 | |
5 mg | In stock | $ 1,800.00 |
Description | Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease. |
In vitro | Cicloprolol, a partial β1-adrenoceptor agonist, is being considered for the treatment of patients with coronary artery disease and impaired left ventricular function[1]. This new β-adrenoceptor partial agonist, Cicloprolol, functions as a β-agonist at normal levels and as a β-antagonist at high levels of adrenergic discharge. The treatment with Cicloprolol is designed to protect the heart against excessive stimulation while maintaining a baseline level of sympathetic drive. Specifically, Cicloprolol exhibits a weak β1-agonistic effect at normal levels of adrenergic discharge and acts as an antagonist at high levels of discharge[2]. |
Molecular Weight | 359.89 |
Formula | C18H30ClNO4 |
CAS No. | 63686-79-3 |
store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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Cicloprolol hydrochloride 63686-79-3 GPCR/G Protein Neuroscience Adrenergic Receptor Cicloprolol Hydrochloride inhibitor inhibit