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Cinacalcet metabolite M4

Catalog No. T10814   CAS 104774-87-0
Synonyms: Rarechem AL BW 1078

Cinacalcet metabolite M4 (Rarechem AL BW 1078) is a metabolite of Cinacalcet. Cinacalcet is an allosteric agonist of Ca receptor.

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Cinacalcet metabolite M4 Chemical Structure
Cinacalcet metabolite M4, CAS 104774-87-0
Pack Size Availability Price/USD Quantity
5 mg In stock $ 50.00
10 mg In stock $ 68.00
25 mg In stock $ 97.00
50 mg In stock $ 139.00
100 mg In stock $ 179.00
200 mg In stock $ 256.00
500 mg In stock $ 384.00
1 mL * 10 mM (in DMSO) In stock $ 47.00
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Purity: 95.28%
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Biological Description
Chemical Properties
Storage & Solubility Information
Description Cinacalcet metabolite M4 (Rarechem AL BW 1078) is a metabolite of Cinacalcet. Cinacalcet is an allosteric agonist of Ca receptor.
Synonyms Rarechem AL BW 1078
Molecular Weight 203.2
Formula C10H12F3N
CAS No. 104774-87-0

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 55 mg/ml (270.67 mM)

TargetMolReferences and Literature

1. Kumar GN, et al. Metabolism and disposition of calcimimetic agent cinacalcet HCl in humans and animalmodels. Drug Metab Dispos. 2004 Dec;32(12):1491-500. 2. Bushinsky DA, et al. Effect of cinacalcet on urine calcium excretion and supersaturation in genetic hypercalciuric stone-forming rats. Kidney Int. 2006 May;69(9):1586-92.

Related compound libraries

This product is contained In the following compound libraries:
Metabolism Compound Library Ion Channel Inhibitor Library

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Keywords

Cinacalcet metabolite M4 104774-87-0 Membrane transporter/Ion channel Metabolism Calcium Channel disease inhibit Drug Metabolite Cinacalcet metabolite M 4 Cinacalcet metabolite M-4 Inhibitor Rarechem AL BW-1078 Rarechem AL BW1078 Rarechem AL BW 1078 metabolism cardiovascular inhibitor

 

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