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Homo-PROTAC pVHL30 degrader 1
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Homo-PROTAC pVHL30 degrader 1
Catalog No. T13722Cas No. 2244684-49-7
Homo-PROTAC pVHL30 degrader 1 is a potent pVHL30 degrader based on PROTAC.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $50 | In Stock | |
| 5 mg | $128 | In Stock | |
| 10 mg | $163 | In Stock | |
| 25 mg | $328 | In Stock | |
| 50 mg | $528 | In Stock | |
| 100 mg | $769 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $198 | In Stock |
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CitedProduct Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | Homo-PROTAC pVHL30 degrader 1 is a potent pVHL30 degrader based on PROTAC. |
| In vitro | Homo-PROTAC pVHL30 degrader 1 dimerizes von Hippel-Lindau (VHL) with high avidity in vitro and induces rapid, potent, and proteasome-dependent self-degradation of VHL in different cell lines, in a highly isoform-selective fashion and without triggering a hypoxic response. |
| Molecular Weight | 1179.45 |
| Formula | C58H82N8O14S2 |
| Cas No. | 2244684-49-7 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 150 mg/mL (127.18 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
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