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IDH1 Inhibitor 2

Catalog No. T11611   CAS 2244895-42-7

IDH1 Inhibitor 2 (compound 13) is a potent IDH1 inhibitor via direct covalent modification of His315 (IC50: 110 nM).

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IDH1 Inhibitor 2 Chemical Structure
IDH1 Inhibitor 2, CAS 2244895-42-7
Pack Size Availability Price/USD Quantity
25 mg 8-10 weeks $ 1,970.00
50 mg 8-10 weeks $ 2,580.00
100 mg 8-10 weeks $ 3,400.00
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This compound is a customized synthesis product. We have a strong synthesis team with excellent synthesis technology and capabilities. However, due to various objective factors, there is a low probability that the synthesis will not be successful. If you need to learn more, please feel free to consult us, we will serve you wholeheartedly.
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Biological Description
Chemical Properties
Storage & Solubility Information
Description IDH1 Inhibitor 2 (compound 13) is a potent IDH1 inhibitor via direct covalent modification of His315 (IC50: 110 nM).
Targets&IC50 IDH1:110 nM
Molecular Weight 406.48
Formula C26H22N4O
CAS No. 2244895-42-7

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

TargetMolReferences and Literature

1. Jakob CG, et al. Novel Modes of Inhibition of Wild-Type Isocitrate Dehydrogenase 1 (IDH1): Direct Covalent Modification of His315. J Med Chem. 2018 Aug 9;61(15):6647-6657.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

IDH1 Inhibitor 2 2244895-42-7 Metabolism Dehydrogenase IDH-1 Inhibitor 2 inhibitor inhibit

 

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