Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty

Kyotorphin acetate

Catalog No. T20172L

Kyotorphin acetate is an endogenous peptide with analgesia activity and can be used as a biomarker of Alzheimer disease.

Kyotorphin acetate

Kyotorphin acetate

Purity: 99.88%
Catalog No. T20172L
Kyotorphin acetate is an endogenous peptide with analgesia activity and can be used as a biomarker of Alzheimer disease.
Pack SizePriceAvailabilityQuantity
1 mg$48In Stock
2 mg$67In Stock
5 mg$95In Stock
10 mg$158In Stock
25 mg$347In Stock
50 mg$519In Stock
100 mg$752In Stock
500 mg$1,570In Stock
1 mL x 10 mM (in DMSO)$142In Stock
Bulk & Custom
Add to Cart
Questions
View More

Related Compound Libraries of "Kyotorphin acetate"

Select Batch
Purity:99.88%
Contact us for more batch information
Resource Download
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Product Introduction

Bioactivity
Description
Kyotorphin acetate is an endogenous peptide with analgesia activity and can be used as a biomarker of Alzheimer disease.
In vitro
The release of immunoreactive Met-enkephalin (I-ME) from the rat striatum was studied in vitro using a batch technique. A basal release of the order of 2-3% of total I-ME tissue content per 10 min was found. Kyotorphin produced dose-dependent I-ME release, with 0.5 mM maximal concentration causing 2-3-fold stimulation of release. This release was calcium-dependent. In concentrations up to 1 mM Kyotorphin did not change the basal release of [3H]noradrenaline, [3H]GABA, [3H]D-aspartate and immunoreactive beta-endorphin from various brain structures[3].
In vivo
Kyotorphin produced a naloxone-reversible potent analgesic effect, yet no inhibitory effect on electrically induced contractions of longitudinal muscle of the guinea pig ileum[1].
Chemical Properties
Molecular Weight397.43
FormulaC17H27N5O6
Storage & Solubility Information
Storagekeep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 65 mg/ml (163.55 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.5162 mL12.5808 mL25.1617 mL125.8083 mL
5 mM0.5032 mL2.5162 mL5.0323 mL25.1617 mL
10 mM0.2516 mL1.2581 mL2.5162 mL12.5808 mL
20 mM0.1258 mL0.6290 mL1.2581 mL6.2904 mL
50 mM0.0503 mL0.2516 mL0.5032 mL2.5162 mL
100 mM0.0252 mL0.1258 mL0.2516 mL1.2581 mL

Calculator

  • Molarity Calculator
  • Dilution Calculator
  • Reconstitution Calculator
  • Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
1 Enter information below:
mg/kg
g
μL
2 Enter the in vivo formulation:
% DMSO
%
%Tween 80
%ddH2O

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

Related Tags: buy Kyotorphin acetate | purchase Kyotorphin acetate | Kyotorphin acetate cost | order Kyotorphin acetate | Kyotorphin acetate chemical structure | Kyotorphin acetate in vivo | Kyotorphin acetate in vitro | Kyotorphin acetate formula | Kyotorphin acetate molecular weight