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Soraprazan
🥰Excellent
Catalog No. T12977Cas No. 261944-46-1
Alias BYK61359, BYK 61359
Soraprazan (BYK61359) is a selective potassium channel inhibitor that inhibits gastric acid secretion and ameliorates age-related eye disease by removing lipofuscin from retinal pigment epithelial (RPE) cells.
Soraprazan
🥰Excellent
Purity: 99.84%
Catalog No. T12977Alias BYK61359, BYK 61359Cas No. 261944-46-1
Soraprazan (BYK61359) is a selective potassium channel inhibitor that inhibits gastric acid secretion and ameliorates age-related eye disease by removing lipofuscin from retinal pigment epithelial (RPE) cells.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 5 mg | $447 | In Stock | |
| 25 mg | $1,530 | In Stock | |
| 50 mg | $1,990 | In Stock | |
| 100 mg | $3,280 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $430 | In Stock |
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Purity:99.84%
ee:99.06%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Soraprazan (BYK61359) is a selective potassium channel inhibitor that inhibits gastric acid secretion and ameliorates age-related eye disease by removing lipofuscin from retinal pigment epithelial (RPE) cells. |
| Targets&IC50 | [14C]AP:0.19 μM, 1 mM potassium ions in ion-loss vesicles:0.1 μM |
| In vitro | Soraprazan is a potent inhibitor of gastric H,K-ATPase, with an IC50 value of 0.1 μM in the presence of 1 mM potassium ions in ion-loss vesicles, and inhibits dibutyryl cyclic AMP-stimulated [14C]AP accumulation in isolated gastric glands with an IC50 value of 0.19 μM. [1] |
| In vivo | Soraprazan 1-27 μmol/kg administered orally showed rapid and stable inhibition of acid secretion in dogs.[1] |
| Alias | BYK61359, BYK 61359 |
| Molecular Weight | 367.44 |
| Formula | C21H25N3O3 |
| Cas No. | 261944-46-1 |
| Smiles | O(CCOC)[C@@H]1C2=C(C=3N(C=C2)C(C)=C(C)N3)N[C@@H]([C@H]1O)C4=CC=CC=C4 |
| Relative Density. | 1.29 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 80 mg/mL (217.72 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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