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[Orn8]-Urotensin II acetate

[Orn8]-Urotensin II acetate is a Urotensin receptor ligand and a partial agonist at Urotensin receptors.

Catalog No. T37527L

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Purity:98.63%

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COA HPLC MS

[Orn8]-Urotensin II acetate

Catalog No. T37527L

[Orn8]-Urotensin II acetate is a Urotensin receptor ligand and a partial agonist at Urotensin receptors.

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Pack Size	Price	Availability
1 mg	$195	In Stock
5 mg	$437	In Stock
10 mg	$646	In Stock
25 mg	$987	In Stock
50 mg	$1,380	In Stock
100 mg	$1,860	In Stock
1 mL x 10 mM (in DMSO)	$928	In Stock

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Product Introduction

Bioactivity

Description	[Orn8]-Urotensin II acetate is a Urotensin receptor ligand and a partial agonist at Urotensin receptors.
Targets&IC50	UT receptor/GPR14:8 (pEC50)
In vivo	[Orn8]-Urotensin II acetate behaves as a full agonist (pEC50 approximately equal 8) at both human and rat UT receptors in the FlipR calcium assay eliciting similar maximal effects as the natural ligand U-II. On the contrary, in the rat aorta bioassay, [Orn8]-Urotensin II acetate behaves as a competitive and selective antagonist (pA2 = 6.56) showing however a small but consistent residual agonist activity[2].

Chemical Properties

Molecular Weight	1434.59
Formula	C₆₅H₈₇N₁₃O₂₀S₂
Cas No.

Storage & Solubility Information

Storage

keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

Solubility Information

DMSO: 14.35 mg/mL (10 mM)

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	0.6971 mL	3.4853 mL	6.9706 mL	34.8532 mL
5 mM	0.1394 mL	0.6971 mL	1.3941 mL	6.9706 mL
10 mM	0.0697 mL	0.3485 mL	0.6971 mL	3.4853 mL

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Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

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Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

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mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

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