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AMP-PCP disodium
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AMP-PCP disodium
Catalog No. T13547LCas No. 7414-56-4
AMP-PCP disodium is an ATP analogue with binding affinity to the N-terminal domain of Hsp90, with a Kd value of 3.8 μM. The binding of AMP-PCP disodium contributes to the formation of an active homodimer of Hsp90.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $64 | In Stock | |
| 5 mg | $197 | In Stock | |
| 10 mg | $293 | In Stock | |
| 25 mg | $497 | In Stock | |
| 50 mg | $693 | In Stock | |
| 100 mg | $982 | In Stock | |
| 500 mg | $1,960 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | AMP-PCP disodium is an ATP analogue with binding affinity to the N-terminal domain of Hsp90, with a Kd value of 3.8 μM. The binding of AMP-PCP disodium contributes to the formation of an active homodimer of Hsp90. |
| In vitro | Under the promotion of AMP-PCP disodium binding, the formation of Hsp135 active homodimers was enhanced by promoting the characteristic slow-effect conformational exchange of cap region ( A90-G117 ) and surrounding region residues ( A141-A111 ). A total of 90 non-proline residues were identified in the triple-labeled Hsp170 and AMP-PCP binding [ 1 ]. |
| Molecular Weight | 549.17 |
| Formula | C11H16N5Na2O12P3 |
| Cas No. | 7414-56-4 |
| Storage | store at low temperature Powder: -20°C for 3 years | In solvent: -80°C for 1 year | |||||||||||||||||||||||||||||||||||
| Solubility Information | H2O: 80 mg/mL (145.67 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
H2O
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