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Antifungal agent 46
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Catalog No. T74976Cas No. 2842067-19-8
Compound 2f (Antifungal Agent 46) is a potent antifungal that inhibits Ras signaling by targeting protein farnesyltransferase [1].
Antifungal agent 46
Antifungal agent 46
😃Good
Catalog No. T74976Cas No. 2842067-19-8
Compound 2f (Antifungal Agent 46) is a potent antifungal that inhibits Ras signaling by targeting protein farnesyltransferase [1].
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 25 mg | $1,520 | 6-8 weeks | |
| 50 mg | $1,980 | 6-8 weeks | |
| 100 mg | $2,500 | 6-8 weeks |
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Product Introduction
Bioactivity
Chemical Properties
| Description | Compound 2f (Antifungal Agent 46) is a potent antifungal that inhibits Ras signaling by targeting protein farnesyltransferase [1]. |
| In vitro | Antifungal agent 46 (compound 2f) exhibits biofilm inhibitory activity at 12.5 μM, with a minimum inhibitory concentration (MIC) twice that of Amphotericin B [1]. |
| In vivo | Antifungal agent 46 (compound 2f, 0.78 μM) inhibits FTase activity in living organisms [1]. |
| Molecular Weight | 565.43 |
| Formula | C26H28BrF3N4O2 |
| Cas No. | 2842067-19-8 |
Storage & Solubility Information
| Storage | Shipping with blue ice. |
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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