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AT-121 hydrochloride

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Purity:100%

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COA HNMR HPLC LCMS

AT-121 hydrochloride

Catalog No. T39529Cas No. 2099681-71-5

AT-121 hydrochloride is a dual agonist of nociception and mu opioid receptor with Ki values of 3.67 and 16.49 nM, respectively.AT-121 hydrochloride is a safe, non-addictive, pain relieving compound with anti-injury and analgesic activity. AT-121 hydrochloride is a safe, non-addictive, pain relieving compound with anti-injury and analgesic activity.

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Pack Size	Price	Availability
1 mg	$350	In Stock
5 mg	$828	In Stock
10 mg	$1,130	In Stock
25 mg	$1,590	In Stock
50 mg	$1,980	In Stock

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Product Introduction

Bioactivity

Description	AT-121 hydrochloride is a dual agonist of nociception and mu opioid receptor with Ki values of 3.67 and 16.49 nM, respectively.AT-121 hydrochloride is a safe, non-addictive, pain relieving compound with anti-injury and analgesic activity. AT-121 hydrochloride is a safe, non-addictive, pain relieving compound with anti-injury and analgesic activity.
In vivo	AT-121 hydrochloride (0.003-0.03 mg/kg; s.c.; Adult male and female rhesus monkeys) produced antinociceptive effects against an acute noxious stimulus, 50 °C water, in a dose-dependent. Having produces a potent antinociceptive effect.[1]

Chemical Properties

Molecular Weight	499.11
Formula	C24H39ClN4O3S
Cas No.	2099681-71-5

Storage & Solubility Information

Storage

store at low temperature Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 50 mg/mL (100 mM)

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.0036 mL	10.0178 mL	20.0357 mL	100.1783 mL
5 mM	0.4007 mL	2.0036 mL	4.0071 mL	20.0357 mL
10 mM	0.2004 mL	1.0018 mL	2.0036 mL	10.0178 mL
20 mM	0.1002 mL	0.5009 mL	1.0018 mL	5.0089 mL
50 mM	0.0401 mL	0.2004 mL	0.4007 mL	2.0036 mL
100 mM	0.0200 mL	0.1002 mL	0.2004 mL	1.0018 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

Dose Conversion

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc