Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty

Cicloprolol hydrochloride

Catalog No. T10812Cas No. 63686-79-3

Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.

Cicloprolol hydrochloride

Cicloprolol hydrochloride

Purity: 97.26%
Catalog No. T10812Cas No. 63686-79-3
Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.
Pack SizePriceAvailabilityQuantity
1 mg$7006-8 weeks
5 mg$1,8006-8 weeks
Bulk & Custom
Add to Cart
Questions
View More
Select Batch
Purity:97.26%
Contact us for more batch information
Resource Download
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Product Introduction

Bioactivity
Description
Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.
In vitro
Cicloprolol, a partial β1-adrenoceptor agonist, is being considered for the treatment of patients with coronary artery disease and impaired left ventricular function[1]. This new β-adrenoceptor partial agonist, Cicloprolol, functions as a β-agonist at normal levels and as a β-antagonist at high levels of adrenergic discharge. The treatment with Cicloprolol is designed to protect the heart against excessive stimulation while maintaining a baseline level of sympathetic drive. Specifically, Cicloprolol exhibits a weak β1-agonistic effect at normal levels of adrenergic discharge and acts as an antagonist at high levels of discharge[2].
Chemical Properties
Molecular Weight359.89
FormulaC18H30ClNO4
Cas No.63686-79-3
Storage & Solubility Information
Storagestore at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

Calculator

  • Molarity Calculator
  • Dilution Calculator
  • Reconstitution Calculator
  • Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
1 Enter information below:
mg/kg
g
μL
2 Enter the in vivo formulation:
% DMSO
%
%Tween 80
%ddH2O

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

Related Tags: buy Cicloprolol hydrochloride | purchase Cicloprolol hydrochloride | Cicloprolol hydrochloride cost | order Cicloprolol hydrochloride | Cicloprolol hydrochloride chemical structure | Cicloprolol hydrochloride in vitro | Cicloprolol hydrochloride formula | Cicloprolol hydrochloride molecular weight