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CP 316311
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CP 316311
Catalog No. T15008Cas No. 175139-41-0
CP 316311 is a specific CRF1 receptor antagonist with potential antidepressant activity and may be used in the study of depression.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $293 | In Stock | |
| 5 mg | $533 | In Stock | |
| 10 mg | $683 | In Stock | |
| 25 mg | $928 | In Stock | |
| 50 mg | $1,260 | In Stock | |
| 100 mg | $1,680 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | CP 316311 is a specific CRF1 receptor antagonist with potential antidepressant activity and may be used in the study of depression. |
| In vitro | CP-316311 is a CRF1 receptor antagonist that completely antagonizes CRF-stimulated adenylyl cyclase activity in rat cortex and endogenously expressed human CRF1 receptors in IMR32 cells[1]. |
| In vivo | CP-316311 (3.2 mg/kg) demonstrates oral efficacy in central nervous system (CNS) models in vivo, blocking the effects of exogenous and endogenous CRF in rodent CNS models[1]. |
| Molecular Weight | 327.46 |
| Formula | C21H29NO2 |
| Cas No. | 175139-41-0 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
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