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CYP1B1-IN-5

CYP1B1-IN-5
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Purity:98.61%
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CYP1B1-IN-5

Catalog No. T73042Cas No. 176442-56-1
CYP1B1-IN-5 is a selective and potent cytochrome P450 1B1 (CYP1B1) inhibitor with an IC50 of 4.7 nM.CYP1B1-IN-5 can be used for the study of metabolism-related diseases.
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Pack SizePriceAvailabilityQuantity
1 mg$195In Stock
5 mg$483In Stock
10 mg$692In Stock
25 mg$1,080In Stock
50 mg$1,490In Stock
100 mg$1,970In Stock
500 mg$3,930In Stock
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Product Introduction

Bioactivity
Description
CYP1B1-IN-5 is a selective and potent cytochrome P450 1B1 (CYP1B1) inhibitor with an IC50 of 4.7 nM.CYP1B1-IN-5 can be used for the study of metabolism-related diseases.
In vitro
CYP1B1-IN-5 (Compound 6q) binds to the binding pocket of CYP1B1 by forming π-π stacking interactions with residues Phe231, Phe134 and heme.[1]
Chemical Properties
Molecular Weight349.12
FormulaC14H8INO2
Cas No.176442-56-1
Storage & Solubility Information
Storage Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Solubility Information
DMSO: 5.63 mg/mL (16.11 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.8643 mL14.3217 mL28.6434 mL143.2172 mL
5 mM0.5729 mL2.8643 mL5.7287 mL28.6434 mL
10 mM0.2864 mL1.4322 mL2.8643 mL14.3217 mL

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