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Enpp-1-IN-14

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Catalog No. T60105Cas No. 2687222-59-7

Enpp-1-IN-14 is a potent inhibitor of Ectonucleotide Pyrophosphatase/Phosphodiesterase-1 (ENPP1) with an IC50 value of 32.38 nM for recombinant human ENPP-1.Enpp-1-IN-14 has anti-tumor activity.

Enpp-1-IN-14

Enpp-1-IN-14

🥰Excellent
Purity: 100%
Catalog No. T60105Cas No. 2687222-59-7
Enpp-1-IN-14 is a potent inhibitor of Ectonucleotide Pyrophosphatase/Phosphodiesterase-1 (ENPP1) with an IC50 value of 32.38 nM for recombinant human ENPP-1.Enpp-1-IN-14 has anti-tumor activity.
Pack SizePriceAvailabilityQuantity
1 mg$51In Stock
5 mg$122In Stock
10 mg$197In Stock
25 mg$455In Stock
50 mg$672In Stock
100 mg$956In Stock
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Purity:100%
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Product Introduction

Bioactivity
Description
Enpp-1-IN-14 is a potent inhibitor of Ectonucleotide Pyrophosphatase/Phosphodiesterase-1 (ENPP1) with an IC50 value of 32.38 nM for recombinant human ENPP-1. Enpp-1-IN-14 has anti-tumor activity.
In vivo
Enpp-1-IN-14 (compound 015) (50 mg/kg; IP; BID, for 31 days) significantly inhibits tumor growth in female C57BL/6 mice (4-6 weeks old) implanted subcutaneously with 2×10^5 MC38 cells.
Chemical Properties
Molecular Weight403.88
FormulaC15H22ClN5O4S
Cas No.2687222-59-7
SmilesCl.COc1cc2ncnc(N3CCCN(CC3)S(N)(=O)=O)c2cc1OC
Relative Density.no data available
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 3.33 mg/mL (8.25 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.4760 mL12.3799 mL24.7598 mL123.7991 mL
5 mM0.4952 mL2.4760 mL4.9520 mL24.7598 mL

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