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hMAO-B-IN-4
🥰Excellent
Catalog No. T67764Cas No. 1666119-75-0
hMAO-B-IN-4 is a selective, reversible and blood–brain barrier (BBB) penetrable inhibitor of human monoamine oxidase-B (hMAO-B, IC50=0.067 μM, Ki= 0.03 μM, hMAO-A, IC50= 33.82 μM).
hMAO-B-IN-4
🥰Excellent
Purity: 99.88%
Catalog No. T67764Cas No. 1666119-75-0
hMAO-B-IN-4 is a selective, reversible and blood–brain barrier (BBB) penetrable inhibitor of human monoamine oxidase-B (hMAO-B, IC50=0.067 μM, Ki= 0.03 μM, hMAO-A, IC50= 33.82 μM).
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 5 mg | $64 | In Stock | |
| 10 mg | $97 | In Stock | |
| 25 mg | $197 | In Stock | |
| 50 mg | $328 | In Stock | |
| 100 mg | $538 | In Stock | |
| 200 mg | $767 | In Stock | |
| 500 mg | $1,150 | In Stock |
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | hMAO-B-IN-4 is a selective, reversible and blood–brain barrier (BBB) penetrable inhibitor of human monoamine oxidase-B (hMAO-B, IC50=0.067 μM, Ki= 0.03 μM, hMAO-A, IC50= 33.82 μM). |
| Targets&IC50 | MAO-A (human):33.82 μM, MAO-B (human):0.03 μM (Ki), MAO-B (human):0.067 μM |
| In vitro | hMAO-B-IN-4 (0-40 μM) shows high selectivity for hMAO-B over hMAO-A, with an SI value of 504.791, and inhibits hMAO-A and hMAO-B with IC50 values of 33.821 μM and 0.067 μM, respectively[1]. |
| Molecular Weight | 320.4 |
| Formula | C20H16O2S |
| Cas No. | 1666119-75-0 |
| Smiles | O=C(\C=C\c1ccc(OCc2ccccc2)cc1)c1cccs1 |
Storage & Solubility Information
| Storage | Shipping with blue ice. | ||||||||||||||||||||
| Solubility Information | DMSO: 3.2 mg/mL (10 mM), Sonication is recommended.  | ||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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