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Lefradafiban

🥰Excellent
Catalog No. T27808Cas No. 149503-79-7
Alias BIBU-104, BIBU104, BIBU 104

Lefradafiban(BIBU-104) is an oral platelet glycoprotein IIb/IIIa receptor antagonist for the study of angina pectoris and acute coronary syndromes.

Lefradafiban

Lefradafiban

🥰Excellent
Purity: 98.37%
Catalog No. T27808Alias BIBU-104, BIBU104, BIBU 104Cas No. 149503-79-7
Lefradafiban(BIBU-104) is an oral platelet glycoprotein IIb/IIIa receptor antagonist for the study of angina pectoris and acute coronary syndromes.
Pack SizePriceAvailabilityQuantity
1 mg$342In Stock
5 mg$828In Stock
10 mg$1,150In Stock
25 mg$1,680In Stock
50 mg$2,290In Stock
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Purity:98.37%
ee:97.87%
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Product Introduction

Bioactivity
Description
Lefradafiban(BIBU-104) is an oral platelet glycoprotein IIb/IIIa receptor antagonist for the study of angina pectoris and acute coronary syndromes.
In vivo
Lefradafiban (30, 45, and 60 mg; oral; three times daily for 48 hours; patients with stable angina undergoing angioplasty) is an effective oral glycoprotein IIb/IIIa receptor blocker.[1]
AliasBIBU-104, BIBU104, BIBU 104
Chemical Properties
Molecular Weight439.46
FormulaC23H25N3O6
Cas No.149503-79-7
SmilesC(NC(OC)=O)(=N)C1=CC=C(C=C1)C2=CC=C(OC[C@@H]3C[C@@H](CC(OC)=O)C(=O)N3)C=C2
Relative Density.1.32g/cm3
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 45 mg/mL (102.4 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.2755 mL11.3776 mL22.7552 mL113.7760 mL
5 mM0.4551 mL2.2755 mL4.5510 mL22.7552 mL
10 mM0.2276 mL1.1378 mL2.2755 mL11.3776 mL
20 mM0.1138 mL0.5689 mL1.1378 mL5.6888 mL
50 mM0.0455 mL0.2276 mL0.4551 mL2.2755 mL
100 mM0.0228 mL0.1138 mL0.2276 mL1.1378 mL

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Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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