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MK-4827 Racemate
🥰Excellent
Catalog No. T22988Cas No. 1038915-75-1
Alias Niraparib Racemate, 2-(4-piperidin-3-ylphenyl)indazole-7-carboxamide
MK-4827 Racemate (Niraparib Racemate) is a selective PARP1 and PARP2 inhibitor with IC50s of 3.8 nM and 2.1 nM, respectively, over 330-fold selectivity for PARP3, V-PARP and Tank1.
MK-4827 Racemate
🥰Excellent
Purity: 99.47%
Catalog No. T22988Alias Niraparib Racemate, 2-(4-piperidin-3-ylphenyl)indazole-7-carboxamideCas No. 1038915-75-1
MK-4827 Racemate (Niraparib Racemate) is a selective PARP1 and PARP2 inhibitor with IC50s of 3.8 nM and 2.1 nM, respectively, over 330-fold selectivity for PARP3, V-PARP and Tank1.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $45 | In Stock | |
| 2 mg | $63 | In Stock | |
| 5 mg | $89 | In Stock | |
| 10 mg | $156 | In Stock | |
| 25 mg | $297 | In Stock | |
| 50 mg | $518 | In Stock | |
| 100 mg | $698 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $121 | In Stock |
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- $55
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Purity:99.47%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | MK-4827 Racemate (Niraparib Racemate) is a selective PARP1 and PARP2 inhibitor with IC50s of 3.8 nM and 2.1 nM, respectively, over 330-fold selectivity for PARP3, V-PARP and Tank1. |
| Targets&IC50 | PARP1:3.8 nM, PARP2:2.1 nM |
| Alias | Niraparib Racemate, 2-(4-piperidin-3-ylphenyl)indazole-7-carboxamide |
| Molecular Weight | 320.39 |
| Formula | C19H20N4O |
| Cas No. | 1038915-75-1 |
| Smiles | NC(=O)c1cccc2cn(nc12)-c1ccc(cc1)C1CCCNC1 |
| Relative Density. | 1.34 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 60 mg/ml (187.27 mM)  | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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