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Senktide acetate
🥰Excellent
Catalog No. T7633L
Alias Senktide acetate(106128-89-6 free base)
Senktide acetate (Senktide acetate(106128-89-6 free base)) is a selective tachykinin NK3 receptor agonist that promotes the consolidation or expression of ELM for the study of Alzheimer's disease.
Senktide acetate
🥰Excellent
Purity: 98.26%
Catalog No. T7633LAlias Senktide acetate(106128-89-6 free base)
Senktide acetate (Senktide acetate(106128-89-6 free base)) is a selective tachykinin NK3 receptor agonist that promotes the consolidation or expression of ELM for the study of Alzheimer's disease.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $82 | In Stock | |
| 5 mg | $189 | In Stock | |
| 10 mg | $283 | In Stock | |
| 25 mg | $479 | In Stock | |
| 50 mg | $686 | In Stock | |
| 100 mg | $997 | In Stock |
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Purity:98.26%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Senktide acetate (Senktide acetate(106128-89-6 free base)) is a selective tachykinin NK3 receptor agonist that promotes the consolidation or expression of ELM for the study of Alzheimer's disease. |
| In vitro | Senktide, as a selective NK3 receptor agonist, excites dopaminergic neurons in the substantia nigra pars compacta in a concentration-dependent manner, with effective concentrations ranging from 3 to 3000 nM. The average EC50 is 41.2±9 nM[1]. |
| In vivo | The locomotor activity induced by the tachykinin NK(3) receptor agonist senktide was characterized. Injection of senktide i.c.v[2]. |
| Alias | Senktide acetate(106128-89-6 free base) |
| Molecular Weight | 902.02 |
| Formula | C42H59N7O13S |
| Smiles | CSCC[C@@H](C(N)=O)NC([C@H](CC(C)C)NC(CNC([C@H](CC1=CC=CC=C1)N(C)C([C@@H](NC([C@H](CC(O)=O)NC(CCC(O)=O)=O)=O)CC2=CC=CC=C2)=O)=O)=O)=O.CC(O)=O |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | store at low temperature,keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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