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UCM-05194
🥰Excellent
Catalog No. T69647Cas No. 2411412-36-5
Alias UCM05194, UCM 05194
UCM-05194 is a selective LPA1 receptor agonist that can improve neuropathic pain and can be used in the study of progressive system diseases.
UCM-05194
🥰Excellent
Catalog No. T69647Alias UCM05194, UCM 05194Cas No. 2411412-36-5
UCM-05194 is a selective LPA1 receptor agonist that can improve neuropathic pain and can be used in the study of progressive system diseases.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $333 | In Stock | |
| 5 mg | $790 | In Stock | |
| 10 mg | $1,120 | In Stock | |
| 25 mg | $1,670 | In Stock | |
| 50 mg | $2,180 | In Stock | |
| 100 mg | $2,930 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
| Description | UCM-05194 is a selective LPA1 receptor agonist that can improve neuropathic pain and can be used in the study of progressive system diseases. |
| In vitro | METHODS: B103 neuroblastoma cells overexpressing LPA1 receptors were seeded (2.5·105 cells) into the upper chamber of a transwell and vehicle (0.1% fatty acid-free bovine serum albumin), LPA 1 μM, or UCM-05194 were added to the lower chamber. After allowing cells to migrate for 5 h, migrated cells were stained with 0.1% crystal violet solution and counted. RESULTS: UCM-05194 induced neurite retraction and UCM-05194 induced cell migration in B103 cells overexpressing LPA1 in the transwell chamber assay. [1] |
| Alias | UCM05194, UCM 05194 |
| Molecular Weight | 465.32 |
| Formula | C19H30BrO6P |
| Cas No. | 2411412-36-5 |
| Smiles | C(CCCCCCCCC(O[C@@H](COP(=O)(O)O)CBr)=O)C1=CC=CC=C1 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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