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Pack Size | Price | Availability | Quantity |
---|---|---|---|
25 mg | $882 | 6-8 weeks | |
50 mg | $1,170 | 6-8 weeks | |
100 mg | $1,770 | 6-8 weeks |
Description | LPA2 antagonist 2 is >480-fold more selective than LPA3 (IC50 of 13.85 μM).LPA2 antagonist 2 is a selective LPA2 antagonist with an IC50 of 28.3 nM and a Ki of 21.1 nM. |
In vitro | Lysophosphatidic acid (LPA) is a phospholipid mediator that elicits a host of biological effects including cell proliferation, survival, motility and differentiation. ?LPA2 antagonist 2 inhibits LPA1 with an Imax of 59.0% at 30 μM[1].?LPA has been shown to regulate cancer cell invasion, metastasis, and resistance to both chemotherapeutics and radiation. |
Molecular Weight | 380.35 |
Formula | C20H16N2O6 |
Cas No. | 36840-10-5 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | |||||||||||||||||||||||||||||||||||
Solubility Information | DMSO: 83.33 mg/mL (219.09 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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