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Pack Size | Price | Availability | Quantity |
---|---|---|---|
2 mg | $34 | In Stock | |
5 mg | $56 | In Stock | |
10 mg | $88 | In Stock | |
25 mg | $173 | In Stock | |
50 mg | $273 | In Stock | |
100 mg | $393 | In Stock | |
200 mg | $559 | In Stock | |
1 mL x 5 mM (in DMSO) | $65 | In Stock |
Description | UNC0321 is an effective inhibitor of histone methyltransferase G9a with a Ki of 63 pM and with IC50s 9 nM and 6 nM in ECSD and CLOT assays. UNC0321 inhibits GLP with IC50s of 15 nM and 23 nM in ECSD and CLOT assays. |
Targets&IC50 | G9a:63 pM (ki), G9a:6-9 nM, GLP:15-23 nM |
In vitro | UNC0321 is inactive against SET7/9, SET8/PreSET7, PRMT3 and JMJD2E[1]. UNC0321 reduces H3K9me2 levels in MDA-MB-231 cells with an IC50 of 11 μM[2]. |
Molecular Weight | 515.69 |
Formula | C27H45N7O3 |
Cas No. | 1238673-32-9 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||
Solubility Information | DMSO: 3.33 mg/ml (6.46 mM), Sonication is recommended. | |||||||||||||||
Solution Preparation Table | ||||||||||||||||
DMSO
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