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Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $54 | In Stock | |
5 mg | $128 | In Stock | |
10 mg | $198 | In Stock | |
25 mg | $397 | In Stock | |
50 mg | $628 | In Stock | |
100 mg | $888 | In Stock | |
500 mg | $1,770 | In Stock | |
1 mL x 10 mM (in DMSO) | $143 | In Stock |
Description | CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptor |
In vitro | CCPA suppressed the mRNA and protein expressions of CnAβ and exerted antihypertrophic effects to a greater degree than CsA. The inhibition of CCPA on cardiomyocyte hypertrophy was counteracted by the A1 receptor antagonist DPCPX[1]. |
In vivo | CCPA (CCPA) was synthesized as a potential high affinity ligand for A1 adenosine receptors. Binding of [3H]PIA to A1 receptors of rat brain membranes was inhibited by CCPA with a Ki-value of 0.4 nM, compared to a Ki-value of 0.8 nM for the parent compound N6-cyclopentyladenosine (CPA)[2]. |
Alias | 2-chloro-N(6)cyclopentyladenosine, 2-CHLORO-N-CYCLOPENTYLADENOSINE |
Molecular Weight | 369.8 |
Formula | C15H20ClN5O4 |
Cas No. | 37739-05-2 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | |||||||||||||||||||||||||||||||||||
Solubility Information | DMSO: 55 mg/ml (148.73 mM) ![]() | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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