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JNJ-DGAT2-A, a specific inhibitor of DGAT2(IC50 = 0.14 μM), can be used in studies about the synthesis of triglycerides.
Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $67 | In Stock | |
5 mg | $163 | In Stock | |
10 mg | $289 | In Stock | |
25 mg | $578 | In Stock | |
50 mg | $833 | In Stock | |
100 mg | $1,150 | In Stock | |
500 mg | $2,290 | In Stock |
Description | JNJ-DGAT2-A, a specific inhibitor of DGAT2(IC50 = 0.14 μM), can be used in studies about the synthesis of triglycerides. |
Targets&IC50 | DGAT-2 (Sf9 insect cell membranes ):0.14 μM |
In vitro | JNJ-DGAT2-A (5 μM) almost completely inhibits the enzymatic activity of recombinant DGAT2 and the DGAT2 activity in HepG2 cell lysates. In HepG2 cells, JNJ-DGAT2-A (0.3125-20 μM) dose-dependently inhibits the generation of TG (50:2), TG (52:2), and TG (54:3) with IC50 values of 0.66, 0.85, and 0.99 μM, respectively[1]. |
Alias | JNJDGAT2A |
Molecular Weight | 523.38 |
Formula | C24H16BrFN4O2S |
Cas No. | 1962931-71-0 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||
Solubility Information | DMSO: 3.0 mg/mL (5.7 mM), Sonication and heating to 60℃ are recommended. | |||||||||||||||
Solution Preparation Table | ||||||||||||||||
DMSO
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