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LP-922761 is a potent, selective, and orally active AAK1 inhibitor with inhibitory effects on BMP-2 induced protein kinase (BIKE).
Pack Size | Price | Availability | Quantity |
---|---|---|---|
2 mg | $76 | In Stock | |
5 mg | $129 | In Stock | |
10 mg | $213 | In Stock | |
25 mg | $382 | In Stock | |
50 mg | $568 | In Stock | |
100 mg | $813 | In Stock |
Description | LP-922761 is a potent, selective, and orally active AAK1 inhibitor with inhibitory effects on BMP-2 induced protein kinase (BIKE). |
Targets&IC50 | BIKE:24 nM, AAK1:7.6 nM (cell assays), AAK1:4.8 nM (enzyme assays) |
In vivo | In mice, the brain-to-plasma ratio of LP-922761 was 0.007, indicating that LP-922761 was basically confined to the peripheral compartment[1]. |
Molecular Weight | 410.47 |
Formula | C21H26N6O3 |
Cas No. | 1454808-95-7 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
Solubility Information | DMSO: 1 mg/ml, Sonication is recommended. |
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