Powder: -20°C for 3 years | In solvent: -80°C for 1 year
OMDM-5 is a potent vanilloid receptor type 1 (TRPV1, EC50 = 75 nM) agonist, showing weak ligand activity at cannabinoid type 1 receptor (CB1, Ki=4.9 μM). OMDM-5 is a selective anandamide cellular uptake (ACU) inhibitor(Ki = 4.8 μM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 148.00 | |
5 mg | In stock | $ 336.00 | |
10 mg | In stock | $ 497.00 | |
25 mg | In stock | $ 793.00 | |
50 mg | In stock | $ 1,130.00 | |
100 mg | In stock | $ 1,520.00 | |
500 mg | In stock | $ 2,970.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 388.00 |
Description | OMDM-5 is a potent vanilloid receptor type 1 (TRPV1, EC50 = 75 nM) agonist, showing weak ligand activity at cannabinoid type 1 receptor (CB1, Ki=4.9 μM). OMDM-5 is a selective anandamide cellular uptake (ACU) inhibitor(Ki = 4.8 μM). |
Targets&IC50 | TRPV1:75 Nm(TRPV1), CB1:4.9 μM(Ki), ACU:4.8 μM(Ki) |
Molecular Weight | 432.64 |
Formula | C26H44N2O3 |
CAS No. | 616884-66-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 65 mg/ml (150.24 mM)
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
OMDM-5 616884-66-3 GPCR/G Protein Membrane transporter/Ion channel Metabolism TRP/TRPV Channel Endogenous Metabolite Cannabinoid Receptor fatty TRP Channel Transient receptor potential channels VR1 FAAH inhibit receptor Inhibitor CB1 vanilloid cells OMDM 5 type CB2 uptake RBL-2H3 acids OMDM5 cannabinoid inhibitor