Powder: -20°C for 3 years | In solvent: -80°C for 1 year
RN-1747 is a selective transient receptor potential cation channel subfamily V member 4 agonists (EC50: hTRPV4 of 0.77 μM, mTRPV4 of 4.0 μM, and rTRPV4 of 4.1 μM). RN-1747 also antagonizes TRPM8 (IC50: 4 μM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
2 mg | In stock | $ 38.00 | |
5 mg | In stock | $ 61.00 | |
10 mg | In stock | $ 116.00 | |
25 mg | In stock | $ 213.00 | |
50 mg | In stock | $ 347.00 | |
100 mg | In stock | $ 555.00 | |
200 mg | In stock | $ 792.00 | |
500 mg | In stock | $ 1,180.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 68.00 |
Description | RN-1747 is a selective transient receptor potential cation channel subfamily V member 4 agonists (EC50: hTRPV4 of 0.77 μM, mTRPV4 of 4.0 μM, and rTRPV4 of 4.1 μM). RN-1747 also antagonizes TRPM8 (IC50: 4 μM). |
Targets&IC50 | hTRPV4:0.77 μM(EC50), TRPM8:4 μM, rTRPV4:4.1 μM(EC50), mTRPV4:4.0 μM(EC50) |
Molecular Weight | 395.86 |
Formula | C17H18ClN3O4S |
CAS No. | 1024448-59-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 75 mg/mL (189.46 mM)
You can also refer to dose conversion for different animals. More
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RN-1747 1024448-59-6 Membrane transporter/Ion channel TRP/TRPV Channel TRP Channel RN1747 Inhibitor Transient receptor potential channels RN 1747 inhibit inhibitor