Shopping Cart
- Remove All
![TargetMol](https://www.targetmol.com/storage/error/oops.webp)
Your shopping cart is currently empty
Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $45 | In Stock | |
2 mg | $81 | In Stock | |
5 mg | $148 | In Stock | |
10 mg | $255 | In Stock | |
25 mg | $536 | In Stock | |
50 mg | $773 | In Stock | |
100 mg | $1,080 | In Stock | |
1 mL x 10 mM (in DMSO) | $163 | In Stock |
Description | UCPH-101 is an inhibitor of excitatory amino acid transporter subtype 1 (EAAT1) with an IC50 of 0.66 μM. |
In vitro | Preincubation with 100 μM UCPH-101 results in a notable reduction in the expression levels of HA-EAAT1 and HA-GLAST. Additionally, UCPH-101 and UCPH-102 exhibit concentration-dependent inhibition of EAAT1 anion currents, with dissociation constant (KD) values of 0.34±0.03 μM (Hill=1.3±0.13, n≥9) for UCPH-101 and 0.17±0.02 μM (Hill=0.97±0.11, n≥7) for UCPH-102. |
Alias | UCPH 101 |
Molecular Weight | 422.48 |
Formula | C27H22N2O3 |
Cas No. | 1118460-77-7 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||
Solubility Information | DMSO: 10.6 mg/mL (25 mM) | |||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||
DMSO
|
Copyright © 2015-2024 TargetMol Chemicals Inc. All Rights Reserved.