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AHR antagonist 2

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Purity:99.12%

ee:100%

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COA LCMS HPLC FNMR HNMR CSFC

AHR antagonist 2

Catalog No. T10269Cas No. 2338747-54-7

AHR antagonist 2 is an antagonist of the aryl hydrocarbon receptor. The IC50s for human AHR and mouse AHR are 0.885 and 2.03 nM, respectively.

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Pack Size	Price	Availability
1 mg	$49	In Stock
5 mg	$118	In Stock
10 mg	$196	In Stock
25 mg	$334	In Stock
50 mg	$472	In Stock
100 mg	$672	In Stock
500 mg	Inquiry	In Stock
1 mL x 10 mM (in DMSO)	$135	In Stock

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Product Introduction

Bioactivity

Description

AHR antagonist 2 is an antagonist of the aryl hydrocarbon receptor. The IC50s for human AHR and mouse AHR are 0.885 and 2.03 nM, respectively.

Chemical Properties

Molecular Weight	418.37
Formula	C20H17F3N4O3
Cas No.	2338747-54-7

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 225.0 mg/mL (537.8 mM)

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.3902 mL	11.9511 mL	23.9023 mL	119.5114 mL
5 mM	0.4780 mL	2.3902 mL	4.7805 mL	23.9023 mL
10 mM	0.2390 mL	1.1951 mL	2.3902 mL	11.9511 mL
20 mM	0.1195 mL	0.5976 mL	1.1951 mL	5.9756 mL
50 mM	0.0478 mL	0.2390 mL	0.4780 mL	2.3902 mL
100 mM	0.0239 mL	0.1195 mL	0.2390 mL	1.1951 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

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A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

Dose Conversion

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