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Bisoprolol hemifumarate
🥰Excellent
Catalog No. T0143Cas No. 104344-23-2
Alias EMD33512, Bisoprolol hemifumarate salt, (±)-Bisoprolol hemifumarate, (±)-Bisoprolol (hemifumarate)
Bisoprolol, a selective beta-1 adrenergic receptor antagonist, selectively and competitively binds to and blocks beta-1 adrenergic receptors in the heart, thereby with antihypertensive activity and devoid of intrinsic sympathomimetic activity.
Bisoprolol hemifumarate
🥰Excellent
Purity: 99.95%
Catalog No. T0143Alias EMD33512, Bisoprolol hemifumarate salt, (±)-Bisoprolol hemifumarate, (±)-Bisoprolol (hemifumarate)Cas No. 104344-23-2
Bisoprolol, a selective beta-1 adrenergic receptor antagonist, selectively and competitively binds to and blocks beta-1 adrenergic receptors in the heart, thereby with antihypertensive activity and devoid of intrinsic sympathomimetic activity.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 25 mg | $30 | In Stock | |
| 50 mg | $46 | In Stock |
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Purity:99.95%
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With extensive experience in compound synthesis, we can provide rapid custom synthesis services for this product according to your research needs.Product Introduction
Bioactivity
Chemical Properties
| Description | Bisoprolol, a selective beta-1 adrenergic receptor antagonist, selectively and competitively binds to and blocks beta-1 adrenergic receptors in the heart, thereby with antihypertensive activity and devoid of intrinsic sympathomimetic activity. |
| Alias | EMD33512, Bisoprolol hemifumarate salt, (±)-Bisoprolol hemifumarate, (±)-Bisoprolol (hemifumarate) |
| Molecular Weight | 383.49 |
| Formula | C20H33NO6 |
| Cas No. | 104344-23-2 |
| Smiles | OC(=O)/C=C/C(=O)O.CC(C)NCC(O)COc1ccc(COCCOC(C)C)cc1.CC(C)NCC(O)COc1ccc(COCCOC(C)C)cc1 |
| Relative Density. | 1.033 g/cm3 |
Storage & Solubility Information
| Storage | keep away from direct sunlight,keep away from moisture,store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 199.3 mM, Sonication is recommended. H2O: 26.08 mM, Sonication is recommended. | ||||||||||||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||||||||||||
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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