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BMS202 hydrochloride (1675203-84-5(free base))
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Purity:99.47%
BMS202 hydrochloride (1675203-84-5(free base))
Catalog No. T4696Cas No. 2089334-95-0
BMS202 hydrochloride (1675203-84-5(free base)) (PD-1/PD-L1 inhibitor 2 hydrochloride) is a small-molecule PD-1/PD-L1 interaction inhibitor (IC50: 18 nM). Biophysical studies demonstrate that BMS202 binds directly to PD-L1. Binding of BMS202 promotes PD-L1 dimerisation and blocks the PD-L1/ PD1 interaction.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $47 | Backorder | |
| 2 mg | $57 | Backorder | |
| 5 mg | $102 | Backorder | |
| 10 mg | $163 | Backorder | |
| 25 mg | $323 | Backorder | |
| 50 mg | $577 | Backorder | |
| 100 mg | $826 | Backorder | |
| 1 mL x 10 mM (in DMSO) | $102 | Backorder |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | BMS202 hydrochloride (1675203-84-5(free base)) (PD-1/PD-L1 inhibitor 2 hydrochloride) is a small-molecule PD-1/PD-L1 interaction inhibitor (IC50: 18 nM). Biophysical studies demonstrate that BMS202 binds directly to PD-L1. Binding of BMS202 promotes PD-L1 dimerisation and blocks the PD-L1/ PD1 interaction. |
| Targets&IC50 | PD-1/PD-L1:18 nM |
| Alias | PD-1/PD-L1 inhibitor 2 hydrochloride |
| Molecular Weight | 455.97 |
| Formula | C25H30ClN3O3 |
| Cas No. | 2089334-95-0 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 30 mg/mL (71.51 mM) | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
DMSO
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